http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020161664-A9

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filingDate 2020-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9b531251e6cba5d3a5d6b6d8544bbcac
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publicationDate 2021-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020161664-A9
titleOfInvention Glucagon-like peptide-1 (glp-1) agonist analog, process of preparation and uses thereof
abstract The present disclosure relates to an analog of glucagon-like peptide-1 (glp-1)receptor agonist. The present disclosure provides analogs of glucagon-like peptide-1 (glp-1) receptor agonist wherein, the amino acid at position 2 of the 5 glucagon-like peptide-1 (glp-1)receptor agonist is replaced with D-Alanine. The analogs of glucagon-like peptide-1 (glp-1) have one or more properties of prolonged half-life, better pharmacokinetic profile, retained biological activity, and being advantageous for relieving the patient's burden by reducing the dosing frequency and dose. The present disclosure further provides processes for 10 preparing synthetic glucagon-like peptide-1 (glp-1) analogs.
priorityDate 2019-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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