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filingDate 2020-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e5d8ad325d7b5f1ced73023fda53e2ed
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publicationDate 2020-07-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020151707-A1
titleOfInvention Novel small molecule cd73 inhibitor, preparation method therefor and pharmaceutical use thereof
abstract The present disclosure relates to a novel small molecule CD73 inhibitor, a preparation method therefor and a pharmaceutical use thereof. Particularly, the present disclosure relates to a small molecule CD73 inhibitor represented by general formula (I), a preparation method therefor, a pharmaceutical composition containing the derivative, and use thereof as a therapeutic agent, particularly in the preparation of a medicament for treating CD73-mediated diseases and conditions. The substituents of general formula (I) are as defined in description.
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priorityDate 2019-01-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023053
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148476559
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419576432
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24664
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21589
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123139311
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21050542
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59149
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89121404
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333634684
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453625151
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID235403547
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID147105327
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023048
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237500907
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6327654
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398081
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454587170
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID878495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023051
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023052
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390906
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8434
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17882607
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023049
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155022836
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023050
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456468049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390905
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2723923
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457633951
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138518252
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426308763
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91043091
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163463895
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419525032
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69926639
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393728
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23959
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID239928908
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228695222
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID344391476
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56318
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VV43
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12040442
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44274198
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733933
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53629922
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141836443
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393672
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62354173
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155023181
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14833043
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393660
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83348
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381477147
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Total number of triples: 381.