http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020063727-A1

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_7a4141a48ff4b100515aaad9e7844563
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14
filingDate 2019-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e92ddf569d38bef9dfe6247ad7373321
publicationDate 2020-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020063727-A1
titleOfInvention Tricyclic ring ask1 inhibitors and use thereof
abstract The present invention relates to a compound as shown in general formula (I), and a pharmaceutically acceptable salt, ester or stereisomer thereof. The present invention also relates to a method for preparing the compound, a pharmaceutic preparation and a pharmaceutical composition comprising the compound. The compound of the present invention can effectively inhibit the amino acid of ASK1 from being phosphorylized, and can inhibit the activation of ASK1. Therefore, the compound can treat and/or prevent diseases mediated by ASK1 and related diseases.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2021031071-A1
priorityDate 2018-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107108519-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019134680-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-101076332-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019200267-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-102482257-A
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423055
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466709409
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468312951
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14049689
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7047
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458397310
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414865104
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2760897
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449170751
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457629025
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408470213
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID75806
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10422
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9956178
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID65239
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454973655
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID75654
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414326734
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425995027
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456171974
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226483970
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27638
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393356
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420942325
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415831477
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399416
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410476576
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID26399
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455346640
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70451296
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411502039
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399415
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409688950
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID26397
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23282906
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226433120
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333721593
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410391573
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457633844
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393278
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333721587
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422032068
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452307770
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458396401
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148775297
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394281
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394485
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152774262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394280
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431923431
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152774261
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395130
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21867666
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID260
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID282842
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501329
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394273
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419512823
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11815320
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457484819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5326161
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8103
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152774263
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559213
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21899815
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414675
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419531804
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53627583
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19995369
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67576
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID80971
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114838927
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458427722
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID416496
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID112706413
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455786159
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78090
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702122
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66582
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413795358
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702142
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421877558
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67749
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394858
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466709418
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467856234
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415831446
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23449475
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226679515
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393355
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67105
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226493567
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312044457
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID150664
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227636051
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6335
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID286883
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415478123
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419571196
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3660089
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455784172
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406035455
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226779200
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226459332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12556661
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419540783
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426208976
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1923
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393726
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467856233
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9251
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID480454
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456413267
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394811
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393714
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403877
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456413165
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559562
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415757485
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419516862
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393917
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7221
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9235
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14917
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409674722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457484625
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID340333809
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24408
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID807
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148821510
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID405930200
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426255796
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419515857
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID405930333
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID83223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450982802
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410531777
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7498
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226526302
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID516039
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409901513
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226754511
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390486
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559516
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70017
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390453
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393661
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426202011
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390484
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31254
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554831
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID313
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5150145
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390485
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457444288
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID303200
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393712
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457623688
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5608
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12554533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456411915
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393705
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412013998
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID149815209
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9233
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13150523
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226645321
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411920046
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453451682
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393636
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81219
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19028163
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21982284
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419556587
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457313432
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136101
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68616177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67517
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457311044
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451518794
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID489547
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID417445
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226582011
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81572838
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468351047
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2774533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226484806
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393638
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226415477
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID468310
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID995
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419549422
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136111

Total number of triples: 221.