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publicationDate 2020-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020014041-A1
titleOfInvention Enzymatic synthesis of 4'-ethynyl nucleoside analogs
abstract The present invention relates to an enzymatic synthesis of 4'-ethynyl-2'-deoxy nucleosides and analogs thereof, for example EFdA, that eliminates the use of protecting groups on the intermediates, improves the stereoselectivity of glycosylation and reduces the number of process steps needed to make said compounds. It also relates to the novel intermediates employed in the process.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5ZV89
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ81EY8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67472
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1256096
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6NJX0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7SH17
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A323
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HL21
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GYW1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83155
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A325
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MGB0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9X8R6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8HYS9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2HPZ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A324
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4L752
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09117
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ18C22
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4J6A8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59635
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID1718
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59602
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO61235
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID40154213
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP12365
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ74IA4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9L9K3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8ZDJ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Y7V3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Y277
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59337
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9DS93
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CDJ0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID53354
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8FYQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8AZH2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID61135779
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ67RZ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO65581
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9KD67
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6J596
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4L415
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9KW87
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6J2J7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3JYQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23072
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59296
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID232449
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9FRP1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6JCG7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ022T0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ88V41
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9E8I5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HM84
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62839
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2S2L2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3MFX2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23071
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8G9H6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23070
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HM97
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9E4U5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4QL95
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0KVG7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6TRU6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4EZD9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CJT2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2RLG9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ944G9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2J068
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO68146
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ895N2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9N0I2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VPK9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4UNB0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP84722
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XHH3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9X795
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5Z4R3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59714
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3A247
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5WEY6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO66540
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3QGT3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MUW7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9X576
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9EV50
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7K8P2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5C8D9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SSM8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5953581
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02HZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01517
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5IKE7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01516
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4QHF4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9M9S1
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID419015
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5D683
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8F3X9

Total number of triples: 1671.