http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019147783-A1

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filingDate 2019-01-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019147783-A1
titleOfInvention Sulfonamide derivatives for protein degradation
abstract DCAF15 is a substrate recognition (adaptor) protein of E3 ubiquitin ligase. Disclosed herein are compounds that recruit ubiquitin ligase CRL4DCAF15, to a target RNA recognition motif (RRM), causing its degradation. Also disclosed herein are compositions and methods of use in treating associated disorders and diseases.
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Total number of triples: 681.