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publicationDate 2019-06-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019126431-A1
titleOfInvention DIARYL SUBSTITUTED 5,5-FUSED RING COMPOUNDS AS C5aR INHIBITORS
abstract The present disclosure provides, inter alia, Compounds of Formula (I) or pharmaceutically acceptable salts thereof that are modulators of the C5a receptor. Also provided are pharmaceutical compositions and methods of use including the treatment of diseases or disorders involving pathologic activation from C5a and non-pharmaceutical applications.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8Y4A7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C8I6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4UYK8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392881
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546247
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6809
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311066
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396842
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8CRM9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID73940242
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6DN04
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451339314
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID824761
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78210
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4331085
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100135489
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID21947
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID104625
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426240855
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29385
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2YUN4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4TMJ3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID379992
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12766
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12765
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8D8R2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12768
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97513
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID50798
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP57926
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12767
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35422
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID41957
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454973655
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12772
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16132265
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100126739
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12771
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419518689
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5291
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CQF3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CXF9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID40848
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81881
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4ZSW0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451046756
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5865
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JJY9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO96720
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60463
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7852
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID514803
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92N38
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8053
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ38WJ3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20699
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID66939874
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID837968
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8FID5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2736281
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LAG4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID42453
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6L6X6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419530079
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00751
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918486
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1232
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08333
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12774
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID42549
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2RJJ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10052
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08505
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60923442
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12775
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1230
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12778
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581812
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7FG96
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID405770
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6KH30
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05880
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A5G4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581866
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05879
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419513998
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01317
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1231
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ16653
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID40904
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01316
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3558
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01320
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01319
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415429153
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8871
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280858
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11949597
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281732
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01321
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63103
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01330
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1234
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281736
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01328
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08317
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51749
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11587
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419576644
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04186
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43919
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID76282
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID37888
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02960
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6MHW4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456636612
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04407
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3LNA1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57007
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01315
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LT81
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID33501
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415728227
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5429
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419529188
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5953011
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5D9N8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1KSQ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0TCP4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852169
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3577
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852088
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ668J9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31ZS8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8624356
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56470774
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3579
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56419405
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ82KI9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100038176
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10296883
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID494186
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01334

Total number of triples: 1435.