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filingDate 2018-12-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019116386-A1
titleOfInvention Oral pharmaceutical compositions of amorphous apremilast and process for preparing thereof
abstract The present invention relates an oral pharmaceutical compositions of Amorphous Apremilast and processes for preparing thereof wherein the core composition comprises: an amorphous form of Apremilast; as an active ingredient, an Ammonio methacrylate copolymer dispersion as a binding agent; a mixture of Lactose monohydrate and corn starch as a diluent; at least one Disintegrant & at least one lubricant and the core is coated with Polyvinyl acetate based film-forming agent; Wherein the said pharmaceutical composition about 90 to 95% of Apremilast is released in about 1 hour in an aqueous buffer solution of about pH 6.8 with a paddle speed of 75 RPM.
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