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publicationDate 2019-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019075259-A1
titleOfInvention MACROCYCLIC COMPOUNDS AS PROTEASE INHIBITORS
abstract The compounds of the present invention are represented by the following compounds having the formula (I) and the formula (I '): in which the substituents R 1 , R 2 , R 2 , R 3 , R 4 , R 5 , R, X, Y and Z are as defined in the description and in which the substituents R 1 , R 2 , R 3 , R 4 , R 5 , R, R, X, Y and Z are as defined in the description. These compounds are used in the treatment of bacterial infections, parasitic infections, fungal infections, cancer, immunological disorders, autoimmune disorders, diseases and neurodegenerative disorders, inflammatory disorders or muscular dystrophy or to ensure immunosuppression for transplanted organs or tissues.
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Total number of triples: 1712.