http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019067498-A2

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filingDate 2018-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_30125397522218f9bb30625a88373a5a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fbc362536118a115adc9b0c495b48ccf
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publicationDate 2019-04-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019067498-A2
titleOfInvention PEPTIDE ANTIBIOTIC COMPLEXES AND METHODS OF USE
abstract The present invention relates to compounds that form covalent bonds with peptidases, the compounds having, in some embodiments, broad-spectrum bioactivity. In various embodiments, the compounds act by inhibiting the bacterial type 1 signal peptidase (SPase), which is an essential protein of these bacteria. The invention also relates to pharmaceutical compositions and methods of treatment using the compounds described in the present invention.
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Total number of triples: 591.