http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2018213219-A1

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filingDate 2018-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c208c83514b1e4c315b529d2ac901f17
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publicationDate 2018-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018213219-A1
titleOfInvention Pyrido[2,3-d]pyrimidin-7ones and related compounds as inhibitors of protein kinases
abstract Identified compounds demonstrate protein kinase inhibitory activity. More specifically, the compounds having the structures below (I) are demonstrated to inhibit receptor interacting kinase 2 (RIPK2) and/or Activin-like kinase 2 (ALK2). Compounds that are either dual RIPK2/ ALK2 inhibitors or that preferentially inhibit RIPK2 or ALK2 could provide therapeutic benefit.
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Total number of triples: 435.