http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2018163190-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a8e8ae0b9179a14cb74b07761a2e089b
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-08
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-08
filingDate 2017-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c548b2551041a1192270734b78b0d599
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fa527e828fb4f067668e430f5d89c6c0
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c030d72cbc8c5dd54c1962d0902c3447
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e557b4e4f83c2dc78159a6f349f7eebb
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_921b34e5834d880022393b3b3933296a
publicationDate 2018-09-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018163190-A1
titleOfInvention An improved process for the preparation of varenicline and salt thereof
abstract of the Invention The present invention relates to an improved process for the preparation of varenicline and salt thereof. The present invention also provides a process for the 2,7preparation of l-(4,5-dinitro-10-aza-tricyclo[6.3.1.0 ]dodeca-2(7),3,5-trien-10-yl)-2,2,2-trifluoroethanone of Formula 4 using ethyl trifluoroacetate and further converted to varenicline and salt thereof.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022035434-A1
priorityDate 2017-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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