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publicationDate 2018-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018009466-A1
titleOfInvention Locked nucleic acid cyclic dinucleotide compounds and uses thereof
abstract The present invention provides highly active locked nucleic acid cyclic -dinucleotide (LNA-CDN) immune stimulators that activate DCs via the cytoplasmic receptor known as STING (Stimulator of Interferon Genes). In particular, the LNA-CDNs of the present invention are provided in the form of a composition comprising one or more cyclic dinucleotides that induce human STING-dependent type I interferon production, wherein the cyclic dinucleotides present in the composition have at least one 2', 4' locked nucleic acids within the cyclic dinucleotide.
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Total number of triples: 2048.