http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2018001973-A1

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filingDate 2017-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d8591510dcbe8e2b56902fad5476104c
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_49adbb32ec9ee616771276115f3af0fe
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publicationDate 2018-01-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018001973-A1
titleOfInvention Pyrazole derivatives having activity against pain
abstract The present invention relates to pyrazole derivatives of formula (I) having pharmacological activity towards the α2δ subunit, in particular the α2δ-1 subunit, of the voltage-gated calcium channel, in particular having dual pharmacological activity towards both the α2δ subunit, in particular the α2δ-1 subunit, of the voltage-gated calcium channel and the μ-opioid receptor. The present invention also relates to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy, in particular for the treatment of pain.
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priorityDate 2016-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 428.