http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017137456-A1

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publicationDate 2017-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2017137456-A1
titleOfInvention Bioconjugates containing sulfamide linkers for use in treatment
abstract The present invention is based on the surprising finding that the linker employed in a bioconjugate, such as an anti-body-drug conjugate, is not therapeutically inert but has an effect on the therapeutic index of the bioconjugate. The present invention thus concerns a method for increasing the therapeutic index of a bioconjugate and the bioconjugates for use in treatment, in particular cancer. The bioconjugates according to the invention have a sulfamide linker comprising a group according to formula (1).
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Total number of triples: 528.