http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017133360-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_e4cd9a2ae528abb61034e08fa7c2d918
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-05
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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J43-00
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filingDate 2016-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c7f9fe88e0df80195acda230ecde0d29
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_da3044eac224813411b3ef868c3e1c9f
publicationDate 2017-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2017133360-A1
titleOfInvention Steroidal compound, composition containing the same and use thereof
abstract Provided in the present invention are a steroidal compound, a composition containing the same and a use thereof. Specifically, disclosed in the present invention are a steroidal compound as shown in formula (I) and a drug composition containing the same, or a crystal form, a pharmaceutically acceptable salt, a hydrate or solvate, a stereoisomer, a prodrug, a metabolite or an isotope variant thereof. The compound according to the present invention can be used as a CYP17 enzyme inhibitor, and has better pharmacokinetic parameters, which can improve drug concentration of the compound in an animal, thereby improving the efficacy and safety of the drug, and in turn the compound may be applied in the preparation of the drug for treating CYP17 enzyme-related diseases (such as prostate cancer).
priorityDate 2016-02-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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