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publicationDate 2017-07-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2017125772-A1
titleOfInvention Baricitinib salts
abstract Novel baricitinib, {1-(ethylsulphonyl)-3-[4-(7 H -pyrrolo[2,3- d ]pirimidin-4-yl)- 1 H -pyrazol-1- yl]azetidin-3-yl}acetonitrile salts are disclosed, that are suitable for use as pharmaceutical active substances. More specifically, salts of baricitinib formed with ethanesulfonic acid, methanesulfonic acid, benzenesulfonic acid, hydrochloric acid, 4-toluenesulfonic acid, oxalic acid, 2-hydroxyethane sulfonic acid, fumaric acid, tartaric acid and cyclamic acid are disclosed.
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priorityDate 2016-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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