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publicationDate 2017-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2017106226-A1
titleOfInvention Hydroxyalkylamine- and hydroxycycloalkylamine-substituted diamine-arylsulfonamide compounds with selective activity in voltage-gated sodium channels
abstract Disclosed are compounds of Formula A, or a salt thereof: Formula (A) wherein R 1 , R 2 , and E are defined herein, which compounds have properties for inhibiting Na v 1.7 ion channels found in peripheral and sympathetic neurons. Also described are pharmaceutical formulations comprising the compounds of Formula A or their salts, and methods of treating pain disorders, cough, and itch using the same.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID129243508
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID340383464
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393605
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID129258431
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419474155
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID520
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395229
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID129249100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419530397
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID340406812
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227338963
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398804
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID340406808
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
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Total number of triples: 646.