http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017042834-A1

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filingDate 2016-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_164bb91a8385a55555e8bbe74b63a585
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publicationDate 2017-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2017042834-A1
titleOfInvention Tricyclic fused pyridin-2-one derivatives and their use as brd4 inhibitors
abstract The present disclosure describes heterocyclic compounds of Formula I or, its stereoisomers, pharmaceutically acceptable salts, complexes, hydrates, solvates, tautomers, polymorphs, racemic mixtures, optically active forms and pharmaceutically active derivatives thereof and pharmaceutical compositions containing them as the active ingredient. The present disclosure also describes the synthesis and characterization of aforementioned compounds to exhibit high anticancer activity. The compounds of the present disclosure are useful as medicaments and their use in the manufacture of medicaments for treatment, prevention, or suppression of diseases, and conditions mediated by one or more BET family of bromodomains.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3539960-A4
priorityDate 2015-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705549
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673022
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126702139
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126702827
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID719710
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID164533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70700318
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456373243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705552
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673023
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126702828
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705593
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID238592305
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705595
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673021
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705556
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407090242
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID293353
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10220139
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705591
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126702140
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395085
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID34796
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705604
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53629107
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433584227
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452280402
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17856120
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705607
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433584234
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126702725
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450514992
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID398459
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456375585
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705597
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3030541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433584223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419563201

Total number of triples: 651.