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publicationNumber WO-2016149668-A1
titleOfInvention Compounds and methods for the enhanced degradation of targeted proteins
abstract The present invention relates to bifunctional compounds, which find utility as modulators of targeted ubiquitination, especially inhibitors of a variety of polypeptides and other proteins which are degraded and/or otherwise inhibited by bifunctional compounds according to the present invention. In particular, the present invention is directed to compounds, which contain on one end a VHL ligand which binds to the ubiquitin ligase and on the other end a moiety which binds a target protein such that the target protein is placed in proximity to the ubiquitin ligase to effect degradation (and inhibition) of that protein. The present invention exhibits a broad range of pharmacological activities associated with compounds according to the present invention, consistent with the degradation/inhibition of targeted polypeptides.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122550988
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID452548
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23668196
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409175
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281095
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504915
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281096
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID464205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226564914
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89689879
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID393516
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493831
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412234809
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535834
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67486
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493848
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67501
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419511170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400331
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536126
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33032
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6646
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395083
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535249
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID231
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25077993
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395166
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408931
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4640
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117719779
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535646
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409994
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2597
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409068
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395130
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID22882
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400140

Total number of triples: 3181.