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publicationDate 2016-09-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016138114-A1
titleOfInvention Therapeutic pyridazine compounds and uses thereof
abstract The present invention relates to compounds of formula (I): (I) and salts thereof, wherein: R 1 -R 4 have any of the values defined in the specification, and compositions and uses thereof. The compounds are useful as inhibitors of BRG1, BRM and/or PB1. Also included are pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various BRG1-mediated disorders, BRM-mediated disorders and/or PB1-mediated disorders.
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Total number of triples: 4561.