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publicationDate 2016-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016106941-A1
titleOfInvention Site-specific polyethylene glycol modified asparaginase, preparation method therefor and application thereof
abstract The present application discloses polyethylene glycol-based asparaginase and application thereof. Polyethylene glycol is coupled to the N-end amino of 1 or 2 subunits of L-asparaginase, and the molecular weight of the polyethylene glycol is 30-40 KDa. The polyethylene glycol is preferably branched and has an aldehyde group serving as an active group. The polyethylene glycol-based asparaginase is suitable for preparing anti-tumor medicaments.
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