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publicationDate 2016-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016086200-A9
titleOfInvention 4,5,6,7-tetrahydro-1 h-pyrazolo[4,3-c]pyridin-3-amine compounds as cbp and/or ep300 inhibitors
abstract The present invention relates to compounds of formula (I) or formula (II): and to salts thereof, wherein R 1 -R 4 of formula (I) and R 1 -R 3 of formula (II) have any of the values defined herein, and compositions and uses thereof. The compounds are useful as inhibitors of CBP and/or EP300. Also included are pharmaceutical compositions comprising a compound of formula (I) of formula (II) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various CBP and/or EP300-mediated disorders.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022072647-A1
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019191667-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11274100-B2
priorityDate 2014-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373580
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766237
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68290
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373579
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT84
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766236
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373578
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT83
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766235
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT80
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID305177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID42607502
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766234
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9909202
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6335613
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766233
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373625
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451114410
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID608099
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766232
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373624
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65064
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766231
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373619
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766229
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419655664
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373618
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XSX5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0G7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766226
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373616
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0G6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766225
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419487788
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419583009
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766223
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID233046
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4386
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373609
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121416972
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766222
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419582883
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373608
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766221
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121373607
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121416970
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID316766220

Total number of triples: 7872.