http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2016058563-A1

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filingDate 2015-10-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f99f4bd8f0f1ce13150bcae3dc2a1b70
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publicationDate 2016-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016058563-A1
titleOfInvention A process for preparing highly pure azilsartan
abstract The present invention relates to a process for preparing 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[ 1,1'-biphenyl]-4-yl]methyl] -2-ethoxy-1H-benzimidazole-7-carboxylic acid of formula (I) (azilsartan). The invention also relates to preparation of new solid forms of intermediates that make it possible to obtain azilsartan with a high purity over 99.7% (HPLC) and to their characterization.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2017131218-A1
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