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publicationDate 2016-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016054445-A1
titleOfInvention Novel cyclic monomer and dimer peptides having integrin antagonist activity
abstract The invention relates to C to N cyclized (C-N cyclic) monomer and dimer peptide molecules, as well as peptide dimers which are connected by linker moieties at the N terminus and the C terminus of each peptide subunit, which inhibit binding of α4β7 to the mucosal addressin cell adhesion molecule (MAdCAM) in vivo, and show high selectivity against α4β1 binding.
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