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publicationDate 2015-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2015023170-A1
titleOfInvention A method for preparation of erlotinib
abstract A method for the preparation N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)- quinazolin-4-amine (erlotinib) from 6,7-bis(2-methoxyethoxy)quinazolin-4(3H)-one and 3-aminophenylacetylene in the presence of titanium(IV) chloride and anisole is reported.
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