http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014160392-A1

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filingDate 2014-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c73c1bf15509a00263a85a41419d7f9b
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publicationDate 2014-10-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2014160392-A1
titleOfInvention Modified docetaxel liposome formulations
abstract The present invention provides compositions for the treatment of cancer. The compositions include liposomes containing a phosphatidylcholine lipid, a sterol, a PEG-lipid, and a taxane. The PEG-lipid constitutes from about 2 to about 8 mol % of the lipids in the liposome. The taxane is docetaxel esterified at the 2'-O position with a heterocyclyl-(C 2-5 alkanoic acid). Methods for preparation of liposomal taxanes and treatment of cancer with liposomal taxanes are also disclosed.
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Total number of triples: 2048.