http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014150173-A1

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filingDate 2014-03-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2014-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2014150173-A1
titleOfInvention Method for identifying inhibitors of protein-protein interaction
abstract A method of using NMR and combinatorial synthesis to identify compounds that bind to a target protein is provided. Embodiments of the present disclosure are directed to methods of making compounds including one or more fragments that bind to a target protein. The target protein may be one which is known to have a binding partner. The compound including one or more fragments that bind to the target protein may be an inhibitor of the binding or other interaction between the target protein and binding partner. According to one aspect, binding fragments are attached to a polypeptide backbone in a conformation which allows binding of the fragments to the target protein.
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