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filingDate 2014-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_755887f9d2a093262d3c0dbd0e8a7a71
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publicationDate 2014-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2014113869-A1
titleOfInvention Processes for the preparation of chiral beta amino acid derivatives using asymmetric hydrogenation catalysts
abstract This invention provides processes for the preparation of Sitagliptin and pharmaceutically acceptable salts thereof, said processes comprising enantioselective hydrogenation of a prochiral enamine using chiral ruthenium catalyst.
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