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filingDate 2013-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2662fb48b6fc8ae7a1bfea2b4e448833
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publicationDate 2014-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2014095775-A1
titleOfInvention Bet-protein-inhibiting dihydroquinoxalinones
abstract The invention concerns BET-protein-inhibiting, in particular BRD4-inhibiting, dihydroquinoxalinones of general formula (I), in which A, X, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and n have the meanings given in the description, intermediates for producing the compounds according to the invention, pharmaceutical agents containing the compounds according to the invention, and their prophylactic and therapeutic use in hyperproliferative diseases, in particular tumour diseases. The invention further concerns the use of BET-protein-inhibitors in viral infections, neurodegenerative diseases, inflammatory illnesses, atherosclerotic diseases, and male fertility control.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID322267944
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID107951
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID240474971
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581161
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128792671
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04141
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16130571
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148195
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID129211
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76287915
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24408
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID457193
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2578
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID140374736

Total number of triples: 1895.