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publicationDate 2013-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2013055897-A1
titleOfInvention 8 - carbamoyl - 2 - (2,3- di substituted pyrid - 6 - yl) -1,2,3,4 -tetrahydroisoquinoline derivatives as apoptosis - inducing agents for the treatment of cancer and immune and autoimmune diseases
abstract Disclosed are compounds of formula (I) which inhibit the activity of anti-apoptotic Bcl-xL proteins, compositions containing the compounds and methods of treating diseases during which Bcl-xL proteins are expressed, eg cancer. X is heteroaryl; Y 1 is phenylene or heteroarylene; L 1 is a linker; Y 2 is cycloalkyi, cycloalkenyl, heterocycloalkyl or heterocycloalkenyl; Z 1 is C(0)OR 9 , C(O)NR 10 R 11 , C(0)R 11 , NR 10 C(O)R 11 , etc.
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Total number of triples: 2613.