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filingDate 2012-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_14115e6208558c57f89577bd98c7b1dc
publicationDate 2013-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2013054862-A1
titleOfInvention Polycyclic pyridone derivative having integrase-inhibiting activity
abstract The present invention relates to a compound represented by formula (I-1), formula (I-2), or formula (I-3) having an antiviral effect, or a pharmaceutically acceptable salt thereof, and in further detail, to a pyridone derivative having HIV integrase-inhibiting activity and a drug, particularly an anti-HIV drug, containing the derivative. The compound of the present invention has integrase-inhibiting activity and/or cell propagation-inhibiting activity against a virus, particularly HIV or a resistant virus thereof. Thus, the compound of the present invention is useful in the prevention or treatment of a variety of illnesses and viral infections (such as AIDS) in which integrase plays a role. (Each symbol in the formulas is as defined in the Specification.)
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