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publicationDate 2012-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2012022707-A1
titleOfInvention Substituted heteroaryl spiropyrrolidine mdm2 antagonists
abstract There are provided compounds of the general formula (I) wherein A, B, V, W, R 1 , R 2 , R 3 , R 3 , and R 4 , are as described herein, enantiomers and pharmaceutically acceptable salts thereof, as well as methods for making said compounds and pharmaceutical compositions containing them. The present compounds are useful as anticancer agents, in particular as agents in the therapeutic and/or prophylactic treatment of solid tumors such as for example breast, colon, lung and prostate tumors.
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Total number of triples: 844.