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filingDate 2011-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_87dbbc0686859d0bca0d3ccf2241b5fc
publicationDate 2011-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2011161128-A1
titleOfInvention Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders
abstract The present invention relates to compounds defined by formula I wherein the variables R 1x , R 2x , R 3x , R 4x , R 5x , R 6x , R 7x , R Nx , R 10x , A x , Z x and m are defined as in claim 1, possessing valuable pharmacological activity. Particularly, the compounds are inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 (11beta- HSD1) and thus are suitable for treatment and prevention of diseases which can be influenced by inhibition of this enzyme, such as metabolic diseases, in particular diabetes type 2, obesity, and dyslipidemia.
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Total number of triples: 2651.