http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2011061996-A1
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_67dd1f39f37bac4617e37d6d5c60aa8b http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_4f17880434a6d164920a5ff9fedfa202 |
classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D257-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-10 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D257-04 |
filingDate | 2010-09-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ec4329c8ea3625f9137f72a28db64f97 |
publicationDate | 2011-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | WO-2011061996-A1 |
titleOfInvention | Process for production of biphenyl derivative |
abstract | Disclosed is a process for producing a biaryltetrazole derivative or a salt thereof which is useful as an intermediate for the production of an angiotensin-II receptor antagonist. The process is characterized by comprising: 1) reacting an aryltetrazole derivative represented by general formula [II] with a benzene derivative represented by general formula [III] to produce a compound represented by general formula [IV]; 2) (a) deprotecting the compound represented by general formula [IV] when R 2 in the compound represented by general formula [IV] is a methyl group that is substituted by a hydroxy group protected by a protecting group, or (b) reducing the compound represented by general formula [IV] to produce a compound represented by general formula [V] when the above-mentioned R 2 is a lower alkoxycarbonyl group; and 3) haloganating the compound represented by general formula [IV] when R 2 in the compound represented by general formula [IV] is a methyl group, or halogenating the compound represented by general formula [V] when R 2 in the compound represented by general formula [IV] is a methyl group that is substituted by a hydroxy group protected by a protecting group or a lower alkoxycarbonyl group (in the formulae, each symbol is as defined in the description). |
isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-104583185-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-5925899-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-5881837-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9624181-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014051008-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014034868-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9527821-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013171643-A1 |
priorityDate | 2009-11-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 363.