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filingDate 2010-04-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3236ee85950ec89eb9e9b20c020efc52
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publicationDate 2010-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010125042-A1
titleOfInvention Isoxazole derivatives
abstract The present invention is concerned with novel isoxazole derivatives of formula (I), wherein X, R 1 , R 2 , R 3 , R 4 and R 5 are as described herein, as well as pharmaceutically acceptable salts and esters thereof. The active compounds of the present invention have affinity and selectivity for GABA A α5 receptor. Further the present invention is concerned with the manufacture of the active compounds of formula I, pharmaceutical compositions containing them and their use as medicaments.
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9206160-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020016443-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014001281-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014001282-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9931329-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013120438-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014001278-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014001279-A1
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9475797-B2
priorityDate 2009-04-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458396411
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11718
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID155764
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134664
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7532
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148431
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424603591
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128138055
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3373
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12638758
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81531
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9868
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID586690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID247404563
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23676152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420314932
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID103689
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449102015
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226445872
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127564392
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415809126
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID783
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468020663
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67794
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129149350
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID249243710
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22411348
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409862605
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409862606
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245510940
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457636484
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136387251
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128641745
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245976713
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129212395
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID247953991
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID244679822
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID134359081
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226410725
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7NDN8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID49800976
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151211
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID49800977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID49800978
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128151852
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399539
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID49800979
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID246524515
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409859814
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419604661
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21865305
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393245
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413645827
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393732
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID247583396
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10351697
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468011638
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245739981

Total number of triples: 360.