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filingDate 2010-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_68c61bac2d73eacdbe95a0a4268b2f97
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publicationDate 2010-09-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010097368-A1
titleOfInvention Isoxazole / o-pyridine derivatives with ethyl and ethenyl linker
abstract The present invention is concerned with novel isoxazole-pyridine derivatives of formula I wherein R 1 , R 2 , R 3 and L are as described herein, as well as pharmaceutically acceptable salts and esters thereof. The active compounds of the present invention have affinity and selectivity for GABA A α5 receptor.. Further the present invention is concerned with the manufacture of the active compounds of formula I, pharmaceutical compositions containing them and their use as medicaments.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226554682
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419604661
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7532
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Total number of triples: 358.