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filingDate 2010-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_15749fdba730cff462b7fc004ebec631
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publicationDate 2010-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010085514-A1
titleOfInvention Fluorescence resonance energy transfer assays for sarco/endoplasmic reticulum calcium atpase and phospholamban
abstract Provided herein are methods for identifying molecules capable of modulating SERCA, the SERCA-PLB complex or the microenvironment of the complex. An exemplary assay provided herein is fluorescence resonance energy transfer (FRET). Also provided herein are FRET assays that are optimized for high-throughput screening (HTS) for identifying small molecules that modulate SERCA or the SERCA-PLB complex. Further provided are kits for carrying out said methods for identifying molecules.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10902
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID399259
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27165
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID171548
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27161
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59140
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9R0J8
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415824567
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416522
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397421
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226416521
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YNX6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCG3V226
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416176433
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409680
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22876684
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419568502
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411181230
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID700
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24847920
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419518979
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5RAD2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00974
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397779
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO02367
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450766143
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136039819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12303145
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4324384
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID474584
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6438350
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419568010
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417567
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86348
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18679889
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ669R9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417566
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID363248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9TRY9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID512313
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9MQ82
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136033793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID312
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID108698710
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419556968
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VHN8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID135955727
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226744222
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP85412
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419526255
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1SWB8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25517
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417419
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22629
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87110531
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GRJ1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87059621
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6331297
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87110530
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406715
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447621240
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87059620
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID246348317
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129561421
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406714
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9K9C6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559517
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87059619
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID246328062
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID6239
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521226
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8AKB8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413807576
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6438639
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559506
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID135864362
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID53313
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393705
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419481434
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87059223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419556475
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70753
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9845
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128984259
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127729761
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2875471
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID46931058

Total number of triples: 734.