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filingDate 2009-10-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2010-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010048306-A1
titleOfInvention High-throughput assay for evaluating dipeptidyl peptidase i activity
abstract A method of screening a compound which modulates dipeptidyl peptidase I (DPPI) activities comprises the steps of adding a peptide substrate of DPPI to a reaction mixture which comprises DPPI and a compound, wherein the peptide substrate of DPPI has at least 3 amino acids and binds to a binding site of DPPI in addition to the S 1 -S 2 site; and measuring the molecular weight of the substrate, wherein a change in the molecular weight of the substrate is indicative of the presence of DPPI activity.
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