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publicationDate 2010-04-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010044401-A1
titleOfInvention Morpholinopurine derivative
abstract Disclosed is a novel compound which can inhibit phosphatidylinositol 3-kinase (PI3K) and/or mammalian target of rapamycin (mTOR) and has an anti-tumor activity.  Specifically disclosed is a compound which can inhibit PI3K and/or mTOR, has an anti-tumor activity, and is represented by formula (1) that has various substituents.  [In formula (1), R 1 , R 2 , R 3 , R 4 , R a , R b , R c and X are as defined in the description.]
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Total number of triples: 1208.