http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2010028089-A2

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filingDate 2009-09-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_60d1127a4a0dd224519398fa45740f06
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publicationDate 2010-03-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010028089-A2
titleOfInvention Agents and methods for treatment of pain
abstract The invention provides agents useful for treating pain. An exemplary agent comprises or consists of the a portion of a retroviral Tat protein. One such agent is the peptide Tat-NR2B9c. This peptide has previously been described as an agent for inhibiting damaging effects of stroke and similar conditions via inhibition of PSD95 interactions with NMDA receptors and/or NOS. The present application provides data showing that the Tat- NR2B9c peptides is effective in alleviation of pain. The alleviation of pain can be obtained at a dose of the peptide below the dose required to inhibit PSD-95 interactions with NMDAR or NOS.
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priorityDate 2008-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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