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publicationDate 2010-02-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010016628-A1
titleOfInvention Conjugated suramin amino compounds for medical conditions
abstract A modification of pharmacokinetics of suramin by use of amino compounds in modification of lipophilicity and protein binding characteristics for tackling the physico-chemical properties of suramin that gives it poor distribution in the body; formulating the resulting product in a form that leads to targeting body fluids like the lymphatic system when administered in a specific way; and determining the route of administration that maximizes targeting with a view to reducing the dosage so as to limit toxicity, hence increase tolerance by patient.
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