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publicationDate 2010-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010009402-A2
titleOfInvention Nilotinib intermediates and preparation thereof
abstract Intermediates of Nilotinib were prepared, including, for example, 3-(trifluoromethyl- 5 -(4-methyl- 1 H-imidazole- 1 -yl)-benzeneamine; 3 -(4-(pyridin-3 -yl)pyrimidin-2-ylamino)-4- methylbenzoyl halogen dihydrochloride; and N-(3-Bromo-5-trifluoromethylphenyl)-4- methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzamide. Nilotinib»3HCl and its crystalline forms are also described.
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Total number of triples: 445.