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filingDate 2009-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2010-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2010007604-A2
titleOfInvention Inhalable microparticles, and methods for the production thereof
abstract A microparticle preparation suitable for pulmonary delivery of an active agent comprises solid particles having a three-dimensional matrix structure and an active agent entrapped and dispersed throughout the three dimensional matrix structure. The particles having a Mass Median Aerodynamic Diameter (MMAD) of from 1 to 5μm, and the three-dimensional matrix comprises a cross-linked polymer susceptible to degradation by human neutrophil elastase. The three dimensional matrix may comprise an interpenetrating network of a polymeric protein and a cross-linked polysaccharide polymer. Methods for producing the microparticles are also described.
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