http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2009108364-A2

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filingDate 2009-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1e8bdd039cbcafdf096948b8e7234a89
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publicationDate 2009-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2009108364-A2
titleOfInvention Antagonistic analogues of ghrh
abstract There is provided a novel series of synthetic antagonistic analogues of hGHRH(l- 29)NH 2 (SEQ E) NO: 1). These analogues inhibit the activity of endogenous hGHRH on the pituitary GHRH receptors, and therefore prevent the release of growth hormone. The analogues also inhibit the proliferation of human cancers through a direct effect on the cancer cells. The inhibitory potencies of the new analogues result from replacement of various amino acids.
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Total number of triples: 633.