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filingDate 2009-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_19454ae0644418f272c019d8dc432e58
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publicationDate 2009-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2009105023-A1
titleOfInvention Pharmaceutical formulation comprising oxabispidines / 236
abstract The present invention relates to modified release formulations comprising oxapispidines, such as the compound tert-butyl (2- {7- [2- (4-cyano-2-fluorophenoxy) ethyl] -9-oxa-3, 7-diazabicyclo- [3.3.1] non-3-yl} ethyl) carbamate. Said formulations are preferably in the form of multiple unit systems providing for an immediate release of drug in combination with an extended release of drug during a period of time of up to 24 hours. The compositions are useful in the treatment of cardiac arrhythmias and additionally providing the possibility for early detection of patients responding with an unfavourable QT prolongation.
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priorityDate 2008-02-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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