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publicationDate 2009-10-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2009094569-A3
titleOfInvention Method for the enzymatic kinetic resolution of acyloxyalkyl thiocarbonates used for the synthesis of acyloxyalkyl carbamates
abstract Methods of enzymatically resolving acyloxyalkyl thiocarbonates useful in the synthesis of acyloxyalkyl carbamates are disclosed. These carbamates can be coupled to drugs containing amines such as R-baclofen or S-pregabalin.
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