http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2008148599-A2
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5f9db723f41b9245df17b048ca637ad2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_150d7c8567b14a91af65abd54a06dc98 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_9313f2b71bb9ace2f0c13b0b2ad95af2 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D257-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D257-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-41 |
filingDate | 2008-04-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b171dca9e7306e1f5fcc23409b14304c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_28d762f04e75f1b73f6834e1ca121656 |
publicationDate | 2008-12-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | WO-2008148599-A2 |
titleOfInvention | Process for obtaining a valsartan salt useful for obtaining valsartan |
abstract | The invention relates to a new salt of Valsartan, in particular to the high-purity dilithium salt of Valsartan, its polymorphs and solvates or hydrates thereof, useful for obtaining Valsartan with a high yield. The process for obtaining the dilithium salt of Valsartan (I) comprises i) Coupling of the intermediate (II) with the 2-(1H-tetrazole-5-il)-phenylboronic acid of formula (III), wherein said coupling takes place in the presence of a lithium base, and a mixture of water and water-miscible organic solvent and a palladium catalyst, to give the dilithium salt of Valsartan of formula (I). |
priorityDate | 2007-06-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 71.