http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2008088727-A2

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filingDate 2008-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9e1b77582ba23501e0500aec3dc38032
publicationDate 2008-07-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2008088727-A2
titleOfInvention Endothelin receptor antagonists
abstract This invention relates to novel endothelin receptor antagonists of the formula (I), derivatives, acceptable acid addition salts, solvates, hydrates and polymorphs thereof. The invention also provides compositions comprising a compound of this invention and the use of such compositions in methods of treating diseases and conditions that are beneficially treated by compounds that block the endothelin signaling pathway that leads to vasoconstriction and -in particular those diseases or conditions beneficially treated by endothelin receptor antagonists.
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Total number of triples: 596.