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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3dd053c0f0e82dd7d1cb8c1a5a63f07e
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publicationDate 2008-02-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2008016187-A1
titleOfInvention Pladienolide target molecule, compound capable of binding to the target molecule, and screening method for the compound
abstract A method for the determination of the binding activity between a compound of interest and splicing factor 3b (SF3b), comprising the steps of: (a) contacting a labeled pladienolide compound and the compound of interest with a cell or a cell fraction; and (b) determining the distribution of the labeled compound bound. The method enables to screen for a novel active compound capable of acting on (binding to) a pladienolide target molecule or the like.
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