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publicationDate 2007-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2007115808-A1
titleOfInvention Arginine prodrugs with high therapeutic activity
abstract Esters of arginine (L- and/or D- enantiomers) with D-galactose useful as prodrugs are described, possessing a high capacity for penetrating cell membranes and the blood-brain barrier. The esters of the invention, once absorbed, gradually release arginine and ensure prolonged and high levels of the drug, generating a substantial and extended therapeutic response over time.
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